SCHEMBL315767

SCHEMBL315767

Cc1nn(-c2ccccc2)nc1C(=O)NC1CCC(c2ccccc2)(N(C)C)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.52
OPRL1 P41146 8/20 0.52
KCNH2 Q12809 2/20 0.47
SCN9A Q15858 2/20 0.47
SCN5A Q14524 1/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
PKM P14618 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
KAT2B Q92831 1/20 0.46
RIPK1 Q13546 1/20 0.45
MAPT P10636 1/20 0.44
POLB P06746 2/20 0.44
HDAC1 Q13547 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL316061 0.99 OPRM1 (0.54) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316094 0.82 KCNH2 (0.49) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316320 0.82 KCNH2 (0.46) OPRM1KCNH2SCN9ASCN5AKDM4E
SCHEMBL315123 0.81 KCNH2 (0.45) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316217 0.80 KCNH2 (0.47) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316450 0.80 KCNH2 (0.47) KCNH2SCN9ASCN5AKDM4ELMNA
SCHEMBL316216 0.79 KCNH2 (0.46) KCNH2SCN9ASCN5AKDM4ELMNA
SCHEMBL316331 0.79 KCNH2 (0.46) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316308 0.79 KCNH2 (0.46) OPRM1OPRL1KCNH2SCN9ASCN5A
SCHEMBL316174 0.78 KCNH2 (0.47) OPRM1OPRL1KCNH2SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed