SCHEMBL316174

SCHEMBL316174

Cc1cccc(CC2(N(C)C)CCC(NC(=O)c3nn(-c4ccccc4)nc3C)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.47
SCN9A Q15858 3/20 0.47
SCN5A Q14524 2/20 0.47
SSTR1 P30872 1/20 0.42
SSTR4 P31391 1/20 0.42
HDAC1 Q13547 1/20 0.41
RIPK1 Q13546 1/20 0.41
POLB P06746 1/20 0.40
OPRK1 P41145 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ADORA2A P29274 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
PKM P14618 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
KAT2B Q92831 1/20 0.39
DRD4 P21917 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316094 0.93 KCNH2 (0.49) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316416 0.91 KCNH2 (0.46) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL317313 0.91 PKM (0.47) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316217 0.90 KCNH2 (0.47) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316308 0.86 KCNH2 (0.46) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316331 0.86 KCNH2 (0.46) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL315123 0.85 KCNH2 (0.45) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316450 0.84 KCNH2 (0.47) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL316216 0.83 KCNH2 (0.46) KCNH2SCN9ASCN5AHDAC1RIPK1
SCHEMBL315767 0.78 OPRM1 (0.52) KCNH2SCN9ASCN5AHDAC1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed