SCHEMBL316320

SCHEMBL316320

Cc1nn(-c2ccccc2)nc1C(=O)NC1CCC(c2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.46
SCN9A Q15858 2/20 0.46
SCN5A Q14524 1/20 0.46
POLB P06746 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
PKM P14618 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
KAT2B Q92831 1/20 0.43
RIPK1 Q13546 1/20 0.42
MAPT P10636 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
CYP2B6 P20813 1/20 0.41
SLC6A2 P23975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316608 0.86 ALDH1A1 (0.43) KCNH2SCN9AKDM4EMAPTALDH1A1
SCHEMBL315633 0.84 KCNH2 (0.44) KCNH2SCN9ASCN5APOLBMEN1
SCHEMBL316461 0.84 KCNH2 (0.44) KCNH2SCN9ASCN5APOLBMEN1
SCHEMBL315767 0.82 OPRM1 (0.52) KCNH2SCN9ASCN5APOLBMEN1
Hydrochloric Acid SCHEMBL316061 0.81 OPRM1 (0.54) KCNH2SCN9ASCN5APOLBMEN1
SCHEMBL316094 0.75 KCNH2 (0.49) KCNH2SCN9ASCN5APOLBMEN1
SCHEMBL315123 0.74 KCNH2 (0.45) KCNH2SCN9ASCN5APOLBKDM4E
SCHEMBL5572496 0.73 ALDH1A1 (0.56) KCNH2MAPTGRIN2DGRIN3BCYP2B6
SCHEMBL316450 0.73 KCNH2 (0.47) KCNH2SCN9ASCN5APOLBMEN1
SCHEMBL316217 0.73 KCNH2 (0.47) KCNH2SCN9ASCN5APOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed