SCHEMBL315901

SCHEMBL315901

CN(C)C1(Cc2ccccc2)CCC(NC(=O)c2ccc(-c3cc(C(F)(F)F)n(C)n3)s2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 2/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC1 Q13547 5/20 0.38
HDAC3 O15379 4/20 0.38
HDAC4 P56524 4/20 0.38
HDAC7 Q8WUI4 4/20 0.38
HDAC2 Q92769 4/20 0.38
HDAC10 Q969S8 4/20 0.38
HDAC11 Q96DB2 4/20 0.38
HDAC8 Q9BY41 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL314999 0.93 ALDH1A1 (0.52) ALDH1A1GAAL3MBTL1POLBKDM4E
SCHEMBL315505 0.92 ALDH1A1 (0.49) ALDH1A1GAAL3MBTL1POLB
SCHEMBL316103 0.92 ALDH1A1 (0.51) ALDH1A1GAAL3MBTL1POLBKDM4E
SCHEMBL316601 0.91 ALDH1A1 (0.49) ALDH1A1GAAL3MBTL1POLBKDM4E
SCHEMBL316384 0.90 ALDH1A1 (0.49) ALDH1A1GAAL3MBTL1POLBKDM4E
SCHEMBL1594447 0.77 ALDH1A1 (0.59) ALDH1A1GAAL3MBTL1KDM4ERAB9A
SCHEMBL1593729 0.76 ALDH1A1 (0.55) ALDH1A1GAAL3MBTL1RAB9ANPC1
SCHEMBL1593669 0.75 ALDH1A1 (0.72) ALDH1A1GAAL3MBTL1RAB9ANPC1
SCHEMBL12589547 0.74 ALDH1A1 (0.55) ALDH1A1GAAL3MBTL1POLBKDM4E
SCHEMBL1593697 0.74 ALDH1A1 (0.63) ALDH1A1GAAL3MBTL1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed