SCHEMBL316601

SCHEMBL316601

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)c2ccc(-c3cc(C(F)(F)F)n(C)n3)s2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
AKT3 Q9Y243 1/20 0.39
GAA P10253 2/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
MCHR1 Q99705 1/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AKT1 P31749 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
EPHX2 P34913 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315505 0.92 ALDH1A1 (0.49) ALDH1A1GAAPOLBL3MBTL1AKT1
SCHEMBL316103 0.91 ALDH1A1 (0.51) ALDH1A1MAPK11MAPK14AKT3GAA
SCHEMBL315901 0.91 ALDH1A1 (0.52) ALDH1A1GAAPOLBL3MBTL1MCHR1
SCHEMBL314999 0.87 ALDH1A1 (0.52) ALDH1A1MAPK11MAPK14GAAPOLB
SCHEMBL316384 0.85 ALDH1A1 (0.49) ALDH1A1GAAPOLBL3MBTL1MAPT
SCHEMBL1597145 0.79 ALDH1A1 (0.54) ALDH1A1AKT3GAAPOLBL3MBTL1
SCHEMBL315879 0.72 CCR1 (0.44) ALDH1A1MAPK11MAPK14MAPTDRD2
SCHEMBL12589547 0.71 ALDH1A1 (0.55) ALDH1A1GAAPOLBL3MBTL1AKT1
SCHEMBL12589468 0.71 ALDH1A1 (0.57) ALDH1A1AKT3GAAL3MBTL1MAPT
SCHEMBL2058346 0.71 ALDH1A1 (0.72) ALDH1A1GAAPOLBL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed