SCHEMBL316641

SCHEMBL316641

Cc1onc(-c2ccccc2Cl)c1C(=O)NC1CCC(CCc2ccccc2)(N(C)C)CC1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.65
MAPT P10636 1/20 0.56
MEN1 O00255 1/20 0.54
CYP2C19 P33261 1/20 0.52
LMNA P02545 2/20 0.52
ALDH1A1 P00352 2/20 0.51
TSHR P16473 1/20 0.51
GHSR Q92847 1/20 0.51
GPBAR1 Q8TDU6 2/20 0.49
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316050 0.92 GHSR (0.61) KMT2AMAPTMEN1LMNAALDH1A1
SCHEMBL316155 0.89 KMT2A (0.56) KMT2AMAPTMEN1LMNAALDH1A1
SCHEMBL316325 0.86 KMT2A (0.61) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL315598 0.85 KMT2A (0.62) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL316058 0.84 KMT2A (0.65) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL316068 0.84 KMT2A (0.60) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL314979 0.83 GHSR (0.62) KMT2AMAPTMEN1LMNAALDH1A1
SCHEMBL315482 0.83 KMT2A (0.62) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL315884 0.83 KMT2A (0.70) KMT2AMAPTMEN1CYP2C19LMNA
SCHEMBL5245600 0.82 KMT2A (0.44) KMT2AMAPTMEN1CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed