Butetamate

Butetamate

SCHEMBL317018

CCC(C(=O)OCCN(CC)CC)c1ccccc1.O=C(O)CC(O)(CC(=O)O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACVR1ADORA1ADORA2AADORA2BADORA3ESR1ESR2FLT3GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSC1HRH1HTR7IDH1IDH2IRAK1JAK1JAK2JAK3MEN1OPRM1P2RX3PDE5ASCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASIGMAR1SLC6A2SYKTACR1TOP2ATYK2

The experimentally established mechanism targets of Butetamate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 3/20 0.55
SLC6A2 known ✓ P23975 1/20 0.48
OPRM1 known ✓ P35372 1/20 0.48
KDM4E B2RXH2 6/20 1.00
MAPT P10636 2/20 0.62
LMNA P02545 6/20 0.57
CYP1A2 P05177 5/20 0.57
CYP2D6 P10635 5/20 0.57
CYP3A4 P08684 4/20 0.56
ALDH1A1 P00352 3/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
KMT2A Q03164 4/20 0.55
TP53 P04637 1/20 0.52
CYP2C9 P11712 1/20 0.52
MAPK1 P28482 1/20 0.52
TSHR P16473 2/20 0.52
NFKB1 P19838 1/20 0.52
PMP22 Q01453 1/20 0.52
HIF1A Q16665 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butamirate SCHEMBL636120 0.93 KDM4E (0.88) KDM4EMAPTLMNACYP1A2CYP2D6
Butetamate SCHEMBL1643343 0.88 KDM4E (0.84) KDM4ELMNACYP1A2CYP2D6CYP3A4
Butetamate SCHEMBL8721011 0.84 KDM4E (0.78) KDM4ELMNACYP1A2CYP2D6CYP3A4
SCHEMBL9588277 0.84 KDM4E (0.78) KDM4ELMNACYP1A2CYP2D6CYP3A4
SCHEMBL9588408 0.82 KDM4E (0.76) KDM4ELMNACYP1A2CYP2D6CYP3A4
Oxalic Acid SCHEMBL9589927 0.80 KDM4E (0.72) KDM4ELMNACYP1A2CYP2D6CYP3A4
Butamirate SCHEMBL668881 0.80 KDM4E (1.00) KDM4ELMNACYP1A2CYP2D6CYP3A4
Butetamate SCHEMBL7339744 0.79 KDM4E (0.70) KDM4ELMNACYP1A2CYP2D6CYP3A4
SCHEMBL9325583 0.78 KDM4E (0.64) KDM4EMAPTLMNACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL26100 0.76 CYP3A4 (0.70) KDM4ELMNACYP1A2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026097641-A1 TROPHOBLAST-FREE ONE-STEP METHOD FOR CULTURING TUMOR INFILTRATING LYMPHOCYTES AND USE THEREOF 毕诺济(上海)生物技术有限公司 2026-05-15 WO disclosed
WO-2025098984-A1 COMPOSITE FILM OF POLYETHERSULFONE AND OF PARTICLES OF ZIRCONIUM OXIDE OF FORMULA ZRO2, AND USE THEREOF AS ION-CONDUCTING MEMBRANE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2025-05-15 WO disclosed
US-20210332392-A1 COMPOSITIONS AND METHODS OF USE THEREOF FOR SCANDIUM SEPARATION FROM RARE EARTH CONTAINING MATERIAL U.S. DEPARTMENT OF ENERGY 2021-10-28 US disclosed
WO-2021217148-A1 COMPOSITIONS AND METHODS OF USE THEREOF FOR SCANDIUM SEPARATION FROM RARE EARTH CONTAINING MATERIAL LAWRENCE LIVERMORE NATIONAL SECURITY, LLC (US) 2021-10-28 WO disclosed
EP-1993741-B1 INLINE APPLICATION OF COATINGS COOK MEDICAL TECHNOLOGIES LLC (US) 2014-03-19 EP disclosed
US-8523937-B2 Controlled drug delivery using a zein layer modified with levulinic acid COOK MEDICAL TECHNOLOGIES LLC (US) 2013-09-03 US disclosed
US-8303648-B2 Artificial venous valve containing therapeutic agent COOK MEDICAL TECHNOLOGIES LLC (US) 2012-11-06 US disclosed
US-8092819-B2 Implantable medical device coated with a bioactive agent Cook Medical Technologies LLC. (US) 2012-01-10 US disclosed
US-8024851-B2 Method of producing a radially expandable prosthesis COOK MEDICAL TECHNOLOGIES LLC (US) 2011-09-27 US disclosed
US-7914841-B2 Inline application of coatings COOK MEDICAL TECHNOLOGIES LLC (US) 2011-03-29 US disclosed
US-20070196423-A1 Implantable medical device coatings with biodegradable elastomer and releasable therapeutic agent MED INSTITUTE, INC. (US) 2007-08-23 US disclosed
US-20070182055-A1 Inline application of coatings COOK INCORPORATED (US) 2007-08-09 US disclosed
US-20070043423-A1 Intraluminal device with a hollow structure MED INSTITUTE INC. (US) 2007-02-22 US disclosed
WO-2005082393-A1 STABILIZED FEVERFEW FORMULATIONS SOFT GEL TECHNOLOGIES, INC. (US) 2005-09-09 WO disclosed
US-20050186269-A1 Stabilized feverfew formulations THE CIT GROUP/CREDIT FINANCE, INC. 2005-08-25 US disclosed
EP-0805680-A2 COMBINATIONAL DRUGS FOR TREATING MIGRAINE AND OTHER ILLNESSES, COMPRISING SESQUITERPENE LACTONES AND B-COMPLEX VITAMINS Ashbury Research Corporation (CA) 1997-11-12 EP disclosed
WO-1996022774-A2 COMBINATIONAL DRUGS FOR TREATING MIGRAINE AND OTHER ILLNESSES, COMPRISING SESQUITERPENE LACTONES AND B-COMPLEX VITAMINS ASHBURY RESEARCH CORPORATION (CA) 1996-08-01 WO disclosed
EP-0098041-B1 SESQUITERPENE LACTONES, EXTRACTS CONTAINING THEM, THEIR PREPARATION AND PHARMACEUTICAL USE R.P. SCHERER CORPORATION (US) 1989-08-02 EP disclosed
US-4758433-A Oil extract of Tanacetum parthenium for treating migraine R. P. SCHERER CORP. (US) 1988-07-19 US disclosed
EP-0098041-A2 Sesquiterpene lactones, extracts containing them, their preparation and pharmaceutical use R.P. SCHERER CORPORATION (US) 1984-01-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050186269-A1 Stabilized feverfew formulations HAMP, S100P, PYGB MEN1 124/4885SLC6A2 2856/4885OPRM1 2902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.