SCHEMBL3170897

SCHEMBL3170897

N#Cc1ccccc1N1CCN(C(=O)C2CCCc3sc(N)nc32)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.42
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MC4R P32245 1/20 0.39
DPP4 P27487 1/20 0.38
ADRB3 P13945 1/20 0.37
DRD2 P14416 2/20 0.37
KRAS P01116 1/20 0.37
TACR3 P29371 1/20 0.36
ATM Q13315 1/20 0.36
PHGDH O43175 1/20 0.36
NAMPT P43490 1/20 0.36
MTOR P42345 1/20 0.36
RPTOR Q8N122 1/20 0.36
MLST8 Q9BVC4 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3157437 0.90 GRM5 (0.41) GRM5ALDH1A1HPGDALOX15HTT
SCHEMBL3170303 0.86 SMN1; SMN2 (0.45) ALDH1A1ALOX15SMN1; SMN2TSHR
SCHEMBL3171977 0.84 ALDH1A1 (0.45) ALDH1A1HTTSMN1; SMN2ADRB3TSHR
SCHEMBL3163995 0.80 KDM4E (0.50) ALDH1A1HPGDHTTSMN1; SMN2HSD17B10
SCHEMBL4797943 0.80 ALDH1A1 (0.46) ALDH1A1HPGDALOX15HTTSMN1; SMN2
SCHEMBL3163269 0.80 DRD2 (0.40) GRM5ALDH1A1SMN1; SMN2DRD2DRD4
SCHEMBL3175358 0.79 CHRM1 (0.40) SMN1; SMN2
SCHEMBL3170296 0.77 SMN1; SMN2 (0.43) ALDH1A1ALOX15SMN1; SMN2TSHR
SCHEMBL3167885 0.77 HTT (0.38) HTTADRB3TSHR
SCHEMBL3156925 0.77 MAPT (0.53) ALDH1A1HPGDSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716128-B1 SUBSTITUTED 4,5,6,7-TETRAHYDRO-BENZOTHIAZOL-2-YLAMINE COMPOUNDS GRUENENTHAL GMBH (DE) 2010-03-31 EP claimed