SCHEMBL3184451

SCHEMBL3184451

O=C(NCCNC(=O)C1CCCCC1)C1CCCCC1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.66
EPHX1 P07099 1/20 0.65
HDAC8 Q9BY41 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.57
HSD17B10 Q99714 2/20 0.57
KEAP1 Q14145 1/20 0.56
NFE2L2 Q16236 1/20 0.56
NPC1 O15118 1/20 0.54
PKM P14618 1/20 0.54
EPHX2 P34913 1/20 0.54
RAB9A P51151 1/20 0.54
KMT2A Q03164 2/20 0.51
HPGD P15428 1/20 0.51
MEN1 O00255 1/20 0.51
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CTSK P43235 1/20 0.50
CHRM1 P11229 3/20 0.49
CES2 O00748 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21078257 0.89 NAAA (0.61) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL61529 0.89 NAAA (0.59) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL17172545 0.89 NAAA (0.82) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL1094484 0.88 NAAA (0.54) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL23595437 0.87 NAAA (0.58) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL1740262 0.87 NAAA (0.58) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL61158 0.87 NAAA (0.58) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL23419143 0.87 NAAA (0.58) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL9034554 0.87 NAAA (0.58) NAAAEPHX1HDAC8HDAC6SMN1; SMN2
SCHEMBL517349 0.87 NAAA (0.73) NAAAEPHX1HDAC8HDAC6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7666971-B2 Amide/urea-modified liquid diphenylmethane diisocyanates BAYER MATERIALSCIENCE LLC (US) 2010-02-23 US claimed
US-20080139777-A1 Amide/urea-modified liquid diphenylmethane diisocyanates BAYER MATERIALSCIENCE LLC 2008-06-12 US claimed
WO-2008060454-A2 AMIDE/UREA-MODIFIED LIQUID DIPHENYLMETHANE DIISOCYANATES BAYER MATERIALSCIENCE LLC (US) 2008-05-22 WO claimed
US-7666971-B2 Amide/urea-modified liquid diphenylmethane diisocyanates BAYER MATERIALSCIENCE LLC (US) 2010-02-23 US disclosed
US-20080139777-A1 Amide/urea-modified liquid diphenylmethane diisocyanates BAYER MATERIALSCIENCE LLC 2008-06-12 US disclosed
WO-2008060454-A2 AMIDE/UREA-MODIFIED LIQUID DIPHENYLMETHANE DIISOCYANATES BAYER MATERIALSCIENCE LLC (US) 2008-05-22 WO disclosed