SCHEMBL3189508

SCHEMBL3189508

O=C1C=C2OCOC2=CC1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5158335 0.71 PKM (0.32)
SCHEMBL19140309 0.70
SCHEMBL7471966 0.67 PKM (0.38)
SCHEMBL5861546 0.67
SCHEMBL9899907 0.67 ALDH1A1 (0.35)
SCHEMBL8688750 0.66 CA1 (0.41)
SCHEMBL8261130 0.64
SCHEMBL17988138 0.62
SCHEMBL9743198 0.57
SCHEMBL8660608 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115279744-A Modified thioxanthone photoinitiators 林特弗德有限公司 2022-11-01 CN claimed
US-4755188-A Aqueous composition for oxidative hair coloring containing developer-coupler combination with substituted phenol coupler WELLA AKTIENGESELLSCHAFT (DE) 1988-07-05 US claimed
US-4452603-A OXIDATIVE DYEING WITH 1-(B-HYDROXYALKYL)-2,4-DIAMINOBENZENE AS COUPLER WELLA AKTIENGESELLSCHAFT (DE) 1984-06-05 US claimed
EP-0012965-B1 PRODUCT AND PROCESS FOR DYEING HAIR Wella Aktiengesellschaft (DE) 1982-08-25 EP claimed
US-4321053-A Hair dyeing composition and process WELLA AKTIENGESELLSCHAFT (DE) 1982-03-23 US claimed
WO-1982000092-A1 HAIR COLORATION METHOD AND COMPOSITION THEREFOR KONRAD E 1982-01-21 WO claimed
EP-0043436-A1 Composition and process for dyeing hair Wella Aktiengesellschaft (DE) 1982-01-13 EP claimed
EP-0012965-A1 Product and process for dyeing hair Wella Aktiengesellschaft (DE) 1980-07-09 EP claimed
WO-1980001241-A1 COMPOSITION AND PROCESS FOR HAIR COLOURATION WELLA AG (DE) 1980-06-26 WO claimed
WO-1980000417-A1 PREPARATION FOR HAIR COLORATION WELLA AG (DE) 1980-03-20 WO claimed
US-20150196544-A1 NOVEL BENZO[d][1,3]-DIOXOL DERIVATIVES CONCERT PHARMACEUTICALS, INC. 2015-07-16 US disclosed
US-20140018390-A1 DEUTERATED BENZO[D][1,3]-DIOXOL DERIVATIVES CONCERT PHARMACEUTICALS, INC. (US) 2014-01-16 US disclosed
US-8450492-B2 Deuterated benzo[D][1,3]-dioxol derivatives CONCERT PHARMACEUTICALS, INC. (US) 2013-05-28 US disclosed
EP-1910322-B1 NOVEL DEUTERATED BENZO [D][1,3]-DIOXOL DERIVATIVES AS SEROTONIN REUPTAKE INHIBITORS CONCERT PHARMACEUTICALS INC (US) 2012-09-05 EP disclosed
US-20100222589-A1 DEUTERATED BENZO[D][1,3]-DIOXOL DERIVATIVES CONCERT PHARMACEUTICALS INC. 2010-09-02 US disclosed
WO-1980001241-A1 COMPOSITION AND PROCESS FOR HAIR COLOURATION WELLA AG (DE) 1980-06-26 WO disclosed
WO-1980000417-A1 PREPARATION FOR HAIR COLORATION WELLA AG (DE) 1980-03-20 WO disclosed
WO-1980000417-A1 PREPARATION FOR HAIR COLORATION WELLA AG (DE) 1980-03-20 WO disclosed
EP-0008080-A2 Hair dyeing composition Wella Aktiengesellschaft (DE) 1980-02-20 EP disclosed
EP-0008080-A2 Hair dyeing composition Wella Aktiengesellschaft (DE) 1980-02-20 EP disclosed