SCHEMBL3204292

SCHEMBL3204292

COCCNC(=O)c1cccc(-c2cccc3cc(Cc4cc(Cl)cc(Cl)c4)sc23)c1

nearest known ligand 0.88

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 12/20 0.88
TP53 P04637 2/20 0.43
HPGD P15428 2/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
S1PR4 O95977 3/20 0.40
S1PR5 Q9H228 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3198777 0.94 GPR52 (1.00) GPR52TP53HPGDMAPTKDM4E
SCHEMBL29452903 0.94 GPR52 (1.00) GPR52TP53HPGDMAPTKDM4E
SCHEMBL13489581 0.94 GPR52 (0.81) GPR52TP53HPGDMAPTKDM4E
SCHEMBL3218938 0.89 GPR52 (0.88) GPR52HPGDS1PR4S1PR5
SCHEMBL1853387 0.89 GPR52 (0.79) GPR52TP53HPGDMAPTKDM4E
SCHEMBL1854490 0.87 GPR52 (0.77) GPR52TP53MAPTS1PR4S1PR5
SCHEMBL3221007 0.87 GPR52 (0.71) GPR52TP53HPGDMAPTKDM4E
SCHEMBL1846908 0.87 GPR52 (0.78) GPR52S1PR4S1PR5
SCHEMBL1850205 0.87 GPR52 (0.78) GPR52S1PR4S1PR5
SCHEMBL3210142 0.87 GPR52 (0.87) GPR52TP53HPGDMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100041891-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 US disclosed
US-20100041891-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 US disclosed
US-20100041891-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041891-A1 AMIDE COMPOUND GPR52, GPR132, NR5A2 GPR52 1/4885TP53 3403/4885HPGD 2979/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.