SCHEMBL3204794

SCHEMBL3204794

COC(=O)C#CC(=O)C1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
EPHX1 P07099 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TSHR P16473 2/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RECQL P46063 1/20 0.33
NAAA Q02083 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5042210 0.74 CES2 (0.46) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL17430884 0.74 CES2 (0.46) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL25240690 0.73 CES2 (0.41) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL14336987 0.73 NPSR1 (0.36) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL14336967 0.73 NPSR1 (0.49) SMN1; SMN2EPHX1NPSR1POLBALDH1A1
SCHEMBL25706 0.72 ALDH1A1 (0.44) SMN1; SMN2NPSR1TSHRALDH1A1
SCHEMBL3001721 0.71 NPSR1 (0.33) SMN1; SMN2NPSR1EPHX2
SCHEMBL5045982 0.69 CES2 (0.41) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL8644101 0.69 CES2 (0.41) SMN1; SMN2CES2CES1HDAC8HDAC6
SCHEMBL8650880 0.69 CES2 (0.41) SMN1; SMN2CES2CES1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100048604-A1 Ligands for Aldoketoreductases TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2010-02-25 US disclosed
WO-2006023821-A2 LIGANDS FOR ALDOKETOREDUCTASES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2006-03-02 WO disclosed
EP-0646570-B1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO (JP) 1998-06-24 EP disclosed
US-5488134-A Preparation of compounds of lignan series SHIONOGI & CO., LTD. (JP) 1996-01-30 US disclosed
CN-1109685-A Process for producing lignan compound SHIONOGI & CO (JP) 1995-10-04 CN disclosed
EP-0646570-A1 PROCESS FOR PRODUCING LIGNAN COMPOUND SHIONOGI & CO., LTD. (JP) 1995-04-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048604-A1 Ligands for Aldoketoreductases AKR1C2, AKR1C1, AKR1B1 SMN1; SMN2 2620/4885CES2 933/4885CES1 242/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.