Oxyquinoline

Oxyquinoline

SCHEMBL3211964

CCO.Oc1cccc2cccnc12

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

MMP1MMP13MMP7MMP8polrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Oxyquinoline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP8 known ✓ P22894 1/20 0.50
MMP13 known ✓ P45452 1/20 0.50
TSHR P16473 3/20 0.81
MMP2 P08253 2/20 0.81
METAP2 P50579 2/20 0.81
COMT P21964 2/20 0.81
CHRM1 P11229 1/20 0.81
ADRA1A P35348 1/20 0.81
METAP1 P53582 1/20 0.81
HDAC8 Q9BY41 1/20 0.81
KDM4E B2RXH2 9/20 0.68
ALOX12 P18054 3/20 0.68
LMNA P02545 4/20 0.58
ALDH1A1 P00352 3/20 0.58
MAPT P10636 4/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
TP53 P04637 2/20 0.50
HTT P42858 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TDP1 Q9NUW8 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxyquinoline SCHEMBL28295336 1.00 TSHR (0.81) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL28162650 0.90 TSHR (0.84) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL3899683 0.90 TSHR (0.66) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL27529898 0.90 TSHR (0.91) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL29365411 0.90 TSHR (1.00) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL37189 0.90 TSHR (1.00) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL29716519 0.90 TSHR (1.00) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL253313 0.90 TSHR (1.00) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL10869516 0.88 TSHR (0.88) TSHRMMP2METAP2COMTCHRM1
Oxyquinoline SCHEMBL28038881 0.88 TSHR (0.88) TSHRMMP2METAP2COMTCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117269159-A Method for simultaneously and quantitatively detecting ferrous iron and ferric iron 江苏省疾病预防控制中心(江苏省公共卫生研究院) 2023-12-22 CN claimed
CN-116003423-A Method for synthesizing spiro compound by photocatalysis 广西大学 2023-04-25 CN claimed
CN-115901650-A Method for detecting total amount of guanidines in body fluid of renal failure patient 西安乐析医疗科技有限公司 2023-04-04 CN claimed
CN-109239045-B A kind of molecular engram ratio fluorescent sensor and preparation and application 中国科学院烟台海岸带研究所 2019-03-26 CN claimed
CN-109239045-A A kind of molecular engram ratio fluorescent sensor and preparation and application 中国科学院烟台海岸带研究所 2019-01-18 CN claimed
CN-106589219-A Preparation method for fluorescent hydrotalcite/acrylic resin composite material 咸阳师范学院 2017-04-26 CN claimed
CN-103113879-B Method for coating silicon dioxide on surface of 8-hydroxyquinoline aluminum UNIV TAIYUAN TECHNOLOGY 2015-02-25 CN claimed
CN-103113879-A Method for coating silicon dioxide on surface of 8-hydroxyquinoline aluminum UNIV TAIYUAN TECHNOLOGY 2013-05-22 CN claimed
CN-120847077-A Method for detecting content of aluminum ions in high-absorptivity resin 浙江卫星新材料科技有限公司 2025-10-28 CN disclosed
CN-117269159-A Method for simultaneously and quantitatively detecting ferrous iron and ferric iron 江苏省疾病预防控制中心(江苏省公共卫生研究院) 2023-12-22 CN disclosed
CN-117269159-A Method for simultaneously and quantitatively detecting ferrous iron and ferric iron 江苏省疾病预防控制中心(江苏省公共卫生研究院) 2023-12-22 CN disclosed
CN-116003423-A Method for synthesizing spiro compound by photocatalysis 广西大学 2023-04-25 CN disclosed
CN-115901650-A Method for detecting total amount of guanidines in body fluid of renal failure patient 西安乐析医疗科技有限公司 2023-04-04 CN disclosed
CN-113295744-B Based on CuV2O6And application thereof in arginine detection 广东省科学院测试分析研究所(中国广州分析测试中心) 2022-03-11 CN disclosed
US-20140296251-A1 MULTIFUNCTIONAL QUINOLINE DERIVATIVES AS ANTI-NEURODEGENERATIVE AGENTS Annji Pharmaceutical Co., Ltd. (TW) 2014-10-02 US disclosed
CN-103113879-A Method for coating silicon dioxide on surface of 8-hydroxyquinoline aluminum UNIV TAIYUAN TECHNOLOGY 2013-05-22 CN disclosed
US-20100047352-A1 COMPOSITIONS AND METHODS FOR TREATING EXCESSIVE BLEEDING HEMO NANOSCIENCE, LLC 2010-02-25 US disclosed
EP-1799192-A2 COMPOSITIONS AND METHODS FOR TREATING EXCESSIVE BLEEDING Pronovost, Allan D. (US) 2007-06-27 EP disclosed
US-20060034935-A1 Compositions and methods for treating excessive bleeding HEMO NANOSCIENCE, LLC 2006-02-16 US disclosed
WO-2006012541-A2 COMPOSITIONS AND METHODS FOR TREATING EXCESSIVE BLEEDING EISENSON HENRY (US) 2006-02-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140296251-A1 MULTIFUNCTIONAL QUINOLINE DERIVATIVES AS ANTI-NEURODEGENERATIVE AGENTS NLN, SNCA, CLN6 MMP8 4387/4885MMP13 4193/4885TSHR 4432/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.