SCHEMBL3224461

SCHEMBL3224461

COCc1cc(C(F)(C(F)(F)F)C(F)(F)F)cc(C)c1NC(=O)c1cc(F)c(C#N)c(N)c1F

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 9/20 0.35
HPGD P15428 5/20 0.35
HSD17B10 Q99714 2/20 0.35
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
RXFP1 Q9HBX9 2/20 0.32
MAPT P10636 1/20 0.32
DHODH Q02127 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MAPK1 P28482 1/20 0.31
RCE1 Q9Y256 1/20 0.31
RET P07949 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3222031 0.88 KDM4E (0.35) KDM4EALDH1A1HPGDHSD17B10RXFP1
SCHEMBL3220704 0.86 ALDH1A1 (0.32) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL3208889 0.85 KDM4E (0.35) KDM4EPOLBALDH1A1HPGDHSD17B10
SCHEMBL3218396 0.76 HDAC1 (0.37) KDM4EPOLBALDH1A1HPGDHSD17B10
SCHEMBL3216773 0.76 CYP1A2 (0.37) POLBKMT2AMEN1MAPTDHODH
SCHEMBL13455946 0.76 CYP1A2 (0.34) POLBKMT2AMEN1MAPTDHODH
SCHEMBL13424937 0.73 MAPK10 (0.44) KDM4EALDH1A1HPGDHSD17B10TP53
SCHEMBL3201600 0.73 MEN1 (0.35) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL3224628 0.73 S1PR3 (0.40) KDM4EPOLB
SCHEMBL3212646 0.72 ALDH1A1 (0.39) KDM4EALDH1A1HPGDHSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120556-B1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2016-03-09 EP disclosed
US-8389766-B2 Insecticidal compounds SYNGENTA CROP PROTECTION LLC (US) 2013-03-05 US disclosed
US-20100056639-A1 INSECTICIDAL COMPOUNDS SYNGENTA CROP PROTECTION, INC. (US) 2010-03-04 US disclosed
EP-2120556-A1 INSECTICIDAL COMPOUNDS Syngeta Participations AG (CH) 2009-11-25 EP disclosed
WO-2008074427-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056639-A1 INSECTICIDAL COMPOUNDS ACHE, CHRM1, NIT2 KDM4E 2732/4885POLB 4533/4885ALDH1A1 122/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.