SCHEMBL322447

SCHEMBL322447

CCCn1c(=O)c2cc(C(=O)c3nc(-c4cccc(C(=O)O)c4)c4ccccn34)ccc2n(C)c1=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 12/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
PPARG P37231 3/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADORA3 P0DMS8 1/20 0.39
ADORA1 P30542 1/20 0.39
NPC1 O15118 1/20 0.39
MMP13 P45452 1/20 0.39
SLC22A8 Q8TCC7 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14916441 0.89 HDAC1 (0.44) RORCPPARGMMP13SLC22A8
SCHEMBL15093887 0.88 ALDH1A1 (0.41) RORCALDH1A1HPGDPPARGADORA2A
SCHEMBL322594 0.88 MMP13 (0.46) RORCPPARGMMP13SLC22A8
SCHEMBL14917381 0.87 RORC (0.41) RORCPPARGADORA2BMMP13SLC22A8
SCHEMBL321910 0.87 RORC (0.44) RORCALDH1A1HPGDPPARGRECQL
SCHEMBL15094156 0.87 GRM2 (0.40) RORCPPARGMMP13SLC22A8
SCHEMBL322637 0.86 HDAC1 (0.44) RORCALDH1A1HPGDPPARGADORA2A
SCHEMBL321765 0.85 RORC (0.43) RORCALDH1A1HPGDPPARGADORA2A
SCHEMBL322293 0.85 ALDH1A1 (0.40) RORCALDH1A1HPGDPPARGRECQL
SCHEMBL14916117 0.85 HPGD (0.40) RORCALDH1A1HPGDPPARGADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9452164-B2 Imidazopyridine derivatives, process for preparation thereof and therapeutic use thereof SANOFI (FR) 2016-09-27 US disclosed
EP-2590976-B1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2015-09-16 EP disclosed
US-20140243328-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2014-08-28 US disclosed
US-8759344-B2 Imidazopyridine derivatives, process for preparation thereof and therapeutic use thereof SANOFI (FR) 2014-06-24 US disclosed
EP-2590976-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2013-05-15 EP disclosed
US-20130116250-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2013-05-09 US disclosed
WO-2012004732-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140243328-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND THERAPEUTIC USE THEREOF CCNY, ENY2, PAH RORC 1361/4885ALDH1A1 2306/4885HPGD 630/4885
US-20130116250-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR PREPARATION THEREOF AND THERAPEUTIC USE THEREOF CCNY, ENY2, PAH RORC 1361/4885ALDH1A1 2306/4885HPGD 630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.