SCHEMBL3227142

SCHEMBL3227142

Cc1ccc2c(c1)OC1CCCN1C2=O

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.60
MAOB P27338 8/20 0.43
HTR2C P28335 3/20 0.41
HTR2A P28223 2/20 0.39
HTR2B P41595 2/20 0.39
NPC1 O15118 1/20 0.37
CYP19A1 P11511 1/20 0.36
KMT2A Q03164 2/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19166896 0.89 GRIA1 (0.60) GRIA1MAOBHTR2CHTR2AHTR2B
SCHEMBL8314975 0.83 GRIA1 (0.82) GRIA1KMT2AMAPT
SCHEMBL31562999 0.83 GRIA1 (0.60) GRIA1
SCHEMBL7631933 0.82 GRIA1 (0.56) GRIA1MAOBHTR2CHTR2AHTR2B
SCHEMBL7631937 0.82 GRIA1 (0.56) GRIA1MAOBHTR2CHTR2AHTR2B
SCHEMBL8367555 0.82 GRIA1 (0.80) GRIA1
SCHEMBL13492425 0.81 GRIA1 (0.42) GRIA1MAOBHTR2CHTR2AHTR2B
SCHEMBL5806598 0.79 GRIA1 (0.53) GRIA1HTR2CHTR2AHTR2B
SCHEMBL5806602 0.79 GRIA1 (0.53) GRIA1HTR2CHTR2AHTR2B
SCHEMBL31563001 0.79 GRIA1 (0.58) GRIA1MAOBHTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025079090-A1 SUBSTITUTED 4-HETEROATOM-ISOQUINOLONE COMPOUNDS, PROCESS OF PREPARATION AND APPLICATIONS THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2025-04-17 WO claimed
EP-2114158-B1 3-SUBSTITUTED-[1,2,3]BENZOTRIAZINONE COMPOUNDS FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMA INC (US) 2012-08-08 EP disclosed
US-20100041647-A1 3-Substituted-[1,2,3]-Benzotriazinone compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed
US-20100041647-A1 3-Substituted-[1,2,3]-Benzotriazinone compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed
US-20100041647-A1 3-Substituted-[1,2,3]-Benzotriazinone compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-02-18 US disclosed
US-20080176793-A1 UPREGULATING ACTIVITY OR EXPRESSION OF BDNF TO MITIGATE COGNITIVE IMPAIRMENT IN ASYMPTOMATIC HUNTINGTON'S SUBJECTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-07-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041647-A1 3-Substituted-[1,2,3]-Benzotriazinone compounds for enhancing glutamatergic synaptic responses GRIN1, GRIN3B, GABRE GRIA1 26/4885MAOB 418/4885HTR2C 176/4885
US-20080176793-A1 UPREGULATING ACTIVITY OR EXPRESSION OF BDNF TO MITIGATE COGNITIVE IMPAIRMENT IN ASYMPTOMATIC HUNTINGTON'S SUBJECTS BDNF, HTT, NTRK2 GRIA1 156/4885MAOB 1217/4885HTR2C 196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.