SCHEMBL3227312

SCHEMBL3227312

O=C(C(CCCCOc1cccc(F)c1)n1cncn1)C1(Cl)CC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.35
HTR1A P08908 2/20 0.35
TSHR P16473 1/20 0.34
NR4A2 P43354 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ENPP2 Q13822 1/20 0.32
FFAR1 O14842 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3230952 0.90 HRH3 (0.41) TSHRMAPK1KDM4EALDH1A1
SCHEMBL3264017 0.83 MAPK1 (0.40) TSHRMAPK1CTSBKDM4E
SCHEMBL3235712 0.79 HRH3 (0.41) KDM4E
SCHEMBL3239393 0.77 HRH3 (0.45) KDM4E
SCHEMBL3238154 0.74 MAPK1 (0.38) TSHRMAPK1KDM4EALDH1A1
SCHEMBL3232108 0.72 MAPK1 (0.40) TSHRMAPK1CTSBKDM4EALDH1A1
SCHEMBL28384165 0.70 MAPT (0.44) TSHRKDM4EALDH1A1
SCHEMBL3232029 0.69 MAPK1 (0.46) TSHRMAPK1L3MBTL1KDM4EALDH1A1
SCHEMBL10568398 0.68 MAPT (0.62) TSHRKDM4EALDH1A1
SCHEMBL3236422 0.67 HRH3 (0.40) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010029066-A1 IMIDAZOLE AND TRIAZOLE COMPOUNDS, USE THEREOF AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2010-03-18 WO disclosed