SCHEMBL3230291

SCHEMBL3230291

CCc1cc(Cl)cc(Cl)c1-c1ccnn1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
P2RX7 Q99572 4/20 0.40
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
COMT P21964 1/20 0.37
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
HTT P42858 1/20 0.36
SCN9A Q15858 1/20 0.35
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13675221 0.75 P2RX7 (0.47) ALDH1A1MAPTP2RX7CYP1A2CYP2D6
SCHEMBL13522941 0.70 ALDH1A1 (1.00) ALDH1A1MAPTCYP3A4COMTHTR2A
SCHEMBL8121886 0.68 ALDH1A1 (0.45) ALDH1A1MAPTP2RX7SMN1; SMN2CYP1A2
Benzene SCHEMBL27840008 0.68 ALDH1A1 (0.60) ALDH1A1MAPTHPGDSMN1; SMN2NPSR1
SCHEMBL2640152 0.67 MAPT (0.44) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL21030631 0.67 ALDH1A1 (0.41) ALDH1A1MAPTCYP1A2CYP2D6CYP2C19
SCHEMBL27002310 0.67 ALDH1A1 (0.44) ALDH1A1MAPTSMN1; SMN2COMTSCN9A
SCHEMBL15950989 0.66 COMT (0.60) ALDH1A1MAPTSMN1; SMN2CYP1A2CYP2D6
SCHEMBL26108533 0.66 SCN9A (0.42) ALDH1A1MAPTP2RX7CYP1A2CYP2D6
SCHEMBL17369090 0.65 CYP1A2 (0.53) ALDH1A1MAPTKMT2ASMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015628-A1 PYRAZOLO [5,1-B] OXAZOLE DERIVATIVES AS CRF1 ANTAGONISTS NOVARTIS AG (CH) 2010-02-11 WO disclosed