SCHEMBL3230293

SCHEMBL3230293

Nc1ncccc1NC(=O)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
POLB P06746 2/20 0.56
SHMT2 P34897 1/20 0.55
BACE1 P56817 1/20 0.52
HDAC3 O15379 3/20 0.50
HDAC1 Q13547 3/20 0.50
HDAC2 Q92769 3/20 0.50
LTA4H P09960 1/20 0.50
MAPK14 Q16539 1/20 0.50
PLAU P00749 1/20 0.49
CASP3 P42574 1/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 1/20 0.48
NAMPT P43490 1/20 0.47
MAOB P27338 1/20 0.47
MGLL Q99685 1/20 0.47
CA12 O43570 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13465238 0.87 SHMT2 (0.54) NPC1RAB9APOLBSHMT2BACE1
SCHEMBL7229196 0.84 NPC1 (0.61) NPC1RAB9APOLBPLAUCASP3
SCHEMBL14091122 0.84 CTSK (0.50) NPC1RAB9AHDAC1SMN1; SMN2HDAC4
SCHEMBL3811403 0.84 NPC1 (0.68) NPC1RAB9APOLBHDAC3HDAC1
SCHEMBL12633528 0.83 HDAC1 (0.78) HDAC3HDAC1HDAC2NAMPTKDM1A
SCHEMBL8789037 0.81 HDAC1 (0.62) NPC1RAB9APOLBHDAC3HDAC1
SCHEMBL3105408 0.81 RAB9A (0.60) NPC1RAB9APOLBCASP3SMN1; SMN2
SCHEMBL9686367 0.81 NPC1 (0.57) NPC1RAB9APOLBLTA4HMAPK14
SCHEMBL7981351 0.81 NPC1 (0.56) NPC1RAB9APOLBHDAC3HDAC1
SCHEMBL30006672 0.81 NPC1 (0.56) NPC1RAB9APOLBHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed