SCHEMBL3236146

SCHEMBL3236146

Cc1c(C(=O)O)c2cc(=O)cc(F)c-2cn1C

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
NOTUM Q6P988 1/20 0.31
POLB P06746 1/20 0.30
MAP2K2 P36507 1/20 0.30
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2148965 0.82 HDAC1 (0.31)
SCHEMBL2149678 0.81
SCHEMBL3230025 0.81 PTGDR2 (0.35)
SCHEMBL4316385 0.79 MEN1 (0.43) MEN1KMT2ANOTUM
SCHEMBL2149199 0.79 ALDH1A1 (0.36) MEN1KMT2AL3MBTL1MAP2K2MAP2K1
SCHEMBL2149741 0.79 PTGDR2 (0.35)
SCHEMBL2149083 0.78
SCHEMBL3242739 0.78
SCHEMBL3632665 0.78 ABCB1 (0.50) MEN1KMT2AL3MBTL1NOTUM
SCHEMBL3244707 0.77 KMT2A (0.38) BRD4MEN1KMT2AMAP2K2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO claimed
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed