SCHEMBL3236371

SCHEMBL3236371

Cc1c(C(=O)O)c2cc(=O)ccc-2cn1CC(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 14/20 0.44
GFER P55789 1/20 0.34
BMPR1B O00238 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
LIPG Q9Y5X9 1/20 0.31
RAB9A P51151 1/20 0.31
METAP2 P50579 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3230237 0.81 PTGDR2 (0.32) PTGDR2GFER
SCHEMBL3347259 0.81 PTGDR2 (0.46) PTGDR2
SCHEMBL3243476 0.80 ALDH1A1 (0.36) GFERRAB9A
SCHEMBL3237136 0.80 TYR (0.39) PTGDR2GFER
SCHEMBL3238452 0.79 BRD9 (0.36) GFERACVRL1ACVR1RAB9A
SCHEMBL3239397 0.79 ALDH1A1 (0.40) GFERRAB9A
SCHEMBL3242838 0.79 CASP3 (0.33) GFER
SCHEMBL3232124 0.77 HDAC1 (0.39) GFERRAB9A
SCHEMBL3243756 0.76 BRD4 (0.36) GFERRAB9A
SCHEMBL2311708 0.76 HSP90AA1 (0.35) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO claimed
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed