SCHEMBL3242838

SCHEMBL3242838

CSCCn1cc2ccc(=O)cc-2c(C(=O)O)c1C

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.33
CDK9 P50750 1/20 0.33
CASP7 P55210 1/20 0.33
MAPK1 P28482 1/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
GFER P55789 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237136 0.84 TYR (0.39) HDAC1HDAC6GFER
SCHEMBL3239397 0.82 ALDH1A1 (0.40) CASP3CDK9CASP7HDAC1HDAC6
SCHEMBL3238452 0.82 BRD9 (0.36) HDAC1HDAC6GFER
SCHEMBL3232124 0.81 HDAC1 (0.39) MAPK1HDAC1HDAC6GFER
SCHEMBL3347259 0.80 PTGDR2 (0.46)
SCHEMBL3243476 0.79 ALDH1A1 (0.36) MAPK1GFER
SCHEMBL3236371 0.79 PTGDR2 (0.44) GFER
SCHEMBL3243756 0.78 BRD4 (0.36) GFER
SCHEMBL2311708 0.75 HSP90AA1 (0.35)
SCHEMBL3240963 0.74 LDHA (0.34) GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed