SCHEMBL3237908

SCHEMBL3237908

Cc1c(C(=O)O)c2cc(=O)ccc-2cn1NC(C)(C)C

nearest known ligand 0.30

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
MAPT P10636 1/20 0.30
AHR P35869 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2149035 0.84
SCHEMBL3235804 0.82 LDHA (0.33) NPC1RAB9AMAPTAHRSMN1; SMN2
SCHEMBL3347068 0.81 RAB9A (0.34) NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL3230237 0.80 PTGDR2 (0.32)
SCHEMBL2150027 0.79 NPC1 (0.34) NPC1RAB9A
SCHEMBL3239111 0.78 KDM4E (0.32) SMN1; SMN2
SCHEMBL3243756 0.77 BRD4 (0.36) NPC1RAB9AMAPTAHRSMN1; SMN2
SCHEMBL3240963 0.76 LDHA (0.34) NPC1RAB9AMAPTAHRSMN1; SMN2
SCHEMBL3352258 0.75 NTRK1 (0.39) NPC1RAB9ASMN1; SMN2
SCHEMBL3237805 0.74 PTGDR2 (0.39) NPC1RAB9AMAPTAHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO claimed
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed