SCHEMBL3239111

SCHEMBL3239111

CCCCNn1cc2ccc(=O)cc-2c(C(=O)O)c1C

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HDAC3 O15379 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
NCOR2 Q9Y618 1/20 0.32
HCAR3 P49019 1/20 0.32
RARB P10826 3/20 0.32
ASAH1 Q13510 2/20 0.31
SLC37A4 O43826 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
GFER P55789 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
GAA P10253 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
AGTR1 P30556 1/20 0.30
AGTR2 P50052 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2150027 0.82 NPC1 (0.34) HSD17B10ASAH1
SCHEMBL2149035 0.82
SCHEMBL3230237 0.81 PTGDR2 (0.32) GFER
SCHEMBL3237136 0.79 TYR (0.39) KDM4EHSD17B10HDAC1MEN1KMT2A
SCHEMBL3237908 0.78 NPC1 (0.30) SMN1; SMN2
SCHEMBL3235804 0.78 LDHA (0.33) SMN1; SMN2
SCHEMBL3347068 0.77 RAB9A (0.34) KDM4EALDH1A1MEN1KMT2AGFER
SCHEMBL3243756 0.74 BRD4 (0.36) KDM4EMEN1KMT2AGFERSMN1; SMN2
SCHEMBL3235748 0.73 GFER (0.35) KDM4EHSD17B10ALDH1A1MEN1KMT2A
SCHEMBL3240963 0.72 LDHA (0.34) KDM4EALDH1A1MEN1KMT2AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO claimed
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed