SCHEMBL3241029

SCHEMBL3241029

COC(=O)C1=C(C)Nc2[nH]ncc2C1c1nc(C)cs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
HSD17B10 Q99714 3/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
PDE1C Q14123 3/20 0.39
TSHR P16473 3/20 0.38
BACE1 P56817 2/20 0.38
ABCC4 O15439 1/20 0.37
PLIN1 O60240 1/20 0.37
CACNA1F O60840 1/20 0.37
GMNN O75496 1/20 0.37
KCNK2 O95069 1/20 0.37
ABCB11 O95342 1/20 0.37
GSR P00390 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3001034 0.80 KDM4E (0.39) KDM4EHSD17B10ALDH1A1SMN1; SMN2HTT
SCHEMBL3000677 0.76 KDM4E (0.39) KDM4EHSD17B10ALDH1A1PDE1CTSHR
SCHEMBL6293550 0.74 KDM4E (0.53) KDM4EHSD17B10ALDH1A1SMN1; SMN2HTT
SCHEMBL10658875 0.70 KDM4E (0.52) KDM4EHSD17B10ALDH1A1SMN1; SMN2PDE1C
SCHEMBL10657847 0.70 BACE1 (0.53) KDM4EHSD17B10ALDH1A1SMN1; SMN2PDE1C
SCHEMBL3004313 0.67 ALDH1A1 (0.56) KDM4EHSD17B10ALDH1A1HTTTSHR
SCHEMBL3000827 0.66 PDE1C (0.45) ALDH1A1PDE1CADORA3ADORA2A
SCHEMBL10664613 0.66 ADORA3 (0.46) KDM4EHSD17B10ALDH1A1SMN1; SMN2HTT
SCHEMBL4258340 0.66 BACE1 (0.35) BACE1CACNA1B
SCHEMBL13209900 0.66 ALDH1A1 (0.39) KDM4EHSD17B10ALDH1A1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed