SCHEMBL4258340

SCHEMBL4258340

CC1=C(C(=O)O)C(c2nc(C)cs2)c2c(C)n[nH]c2N1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.35
CACNA1B Q00975 2/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3001034 0.87 KDM4E (0.39) GAA
SCHEMBL3246994 0.76 ALDH1A1 (0.47) GAA
SCHEMBL3241029 0.66 KDM4E (0.39) BACE1CACNA1B
SCHEMBL4253439 0.62 ALDH1A1 (0.59) GAA
SCHEMBL7278444 0.60 CACNA1F (0.39) CACNA1B
SCHEMBL7279849 0.60 CACNA1F (0.39) CACNA1B
SCHEMBL10721351 0.57 DYRK1A (0.34) BACE1CACNA1BGAA
SCHEMBL10375741 0.57 KDM4E (0.38) BACE1CACNA1B
SCHEMBL128971 0.57
SCHEMBL7410687 0.56 CACNA1B (0.61) CACNA1BGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed