SCHEMBL3241492

SCHEMBL3241492

COc1cccc(OCC(=O)Nc2ccc(-c3cn[nH]c3)cc2OCCCN)c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.55
MELK Q14680 1/20 0.53
CDC42BPA Q5VT25 4/20 0.50
ROCK1 Q13464 5/20 0.49
KDM4E B2RXH2 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
TP53 P04637 1/20 0.48
RECQL P46063 1/20 0.48
MAPK10 P53779 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ALDH1A1 P00352 2/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3247042 0.95 ROCK2 (0.56) ROCK2CDC42BPAROCK1KDM4ENPC1
SCHEMBL3247286 0.92 ROCK2 (0.59) ROCK2CDC42BPAROCK1KDM4ENPC1
SCHEMBL3249259 0.92 ROCK2 (0.58) ROCK2CDC42BPAROCK1KDM4ENPC1
SCHEMBL3245748 0.89 ROCK2 (0.70) ROCK2CDC42BPAROCK1
SCHEMBL3129506 0.85 ROCK2 (0.64) ROCK2CDC42BPAROCK1
SCHEMBL3249358 0.83 ROCK2 (0.56) ROCK2CDC42BPAROCK1KMT2AL3MBTL1
SCHEMBL3243858 0.81 ROCK2 (0.53) ROCK2CDC42BPAROCK1NPC1RAB9A
SCHEMBL3241106 0.80 ROCK2 (0.68) ROCK2CDC42BPAROCK1
SCHEMBL3124817 0.80 ROCK2 (0.64) ROCK2CDC42BPAROCK1KMT2A
SCHEMBL3242171 0.79 ROCK2 (0.67) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed