SCHEMBL3249259

SCHEMBL3249259

COc1cccc(OCC(=O)Nc2ccc(-c3cn[nH]c3)cc2OCCO)c1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.58
ROCK1 Q13464 6/20 0.58
CDC42BPA Q5VT25 5/20 0.54
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
KMT2A Q03164 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3247286 0.96 ROCK2 (0.59) ROCK2ROCK1CDC42BPAALDH1A1KDM4E
SCHEMBL3247042 0.93 ROCK2 (0.56) ROCK2ROCK1CDC42BPAALDH1A1KDM4E
SCHEMBL3241492 0.92 ROCK2 (0.55) ROCK2ROCK1CDC42BPAALDH1A1KDM4E
SCHEMBL3245748 0.91 ROCK2 (0.70) ROCK2ROCK1CDC42BPA
SCHEMBL3129506 0.88 ROCK2 (0.64) ROCK2ROCK1CDC42BPA
SCHEMBL3249358 0.86 ROCK2 (0.56) ROCK2ROCK1CDC42BPAKMT2AL3MBTL1
SCHEMBL3243858 0.84 ROCK2 (0.53) ROCK2ROCK1CDC42BPAKMT2ANPC1
SCHEMBL3248264 0.83 ROCK2 (0.62) ROCK2ROCK1CDC42BPANPC1RAB9A
SCHEMBL3245171 0.83 ROCK2 (0.69) ROCK2ROCK1
SCHEMBL3124817 0.82 ROCK2 (0.64) ROCK2ROCK1CDC42BPAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed