SCHEMBL3242147

SCHEMBL3242147

O=C(O)Oc1ccc(C(=O)c2ccc([N+](=O)[O-])cc2F)o1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CES2 O00748 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
MAPT P10636 2/20 0.36
HIF1A Q16665 1/20 0.36
LMNA P02545 3/20 0.35
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240065 0.87 ALDH1A1 (0.38) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL3242146 0.83 ALDH1A1 (0.47) ALDH1A1CYP3A4ALOX15TDP1CES2
SCHEMBL5365803 0.79 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL3241870 0.78 ALDH1A1 (0.40) ALDH1A1KMT2AMEN1MAPTHIF1A
SCHEMBL3239963 0.76 ALDH1A1 (0.43) ALDH1A1ALOX15TDP1CES2KMT2A
SCHEMBL25837924 0.75 ALDH1A1 (0.64) ALDH1A1CYP3A4ALOX15TDP1CES2
SCHEMBL77925 0.75 ALDH1A1 (0.64) ALDH1A1CYP3A4ALOX15TDP1CES2
Hydrochloric Acid SCHEMBL17164230 0.74 ALDH1A1 (0.62) ALDH1A1CYP3A4ALOX15TDP1CES2
SCHEMBL27604207 0.72 CES2 (0.56) ALDH1A1CYP3A4ALOX15TDP1CES2
SCHEMBL28281577 0.70 ALDH1A1 (0.57) ALDH1A1CYP3A4ALOX15TDP1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1418176-B1 Pyrazole derivates, their preparation and their use in drugs SANOFI AVENTIS DEUTSCHLAND (DE) 2010-04-28 EP disclosed
EP-1418176-A1 Pyrazole derivates, their preparation and their use in drugs Aventis Pharma Deutschland GmbH (DE) 2004-05-12 EP disclosed
EP-0908456-B1 Pyrazole derivatives, their preparation and their use in drugs AVENTIS PHARMA GMBH (DE) 2003-12-17 EP disclosed
EP-0908456-A1 Pyrazole derivatives, their preparation and their use in drugs Hoechst Marion Roussel Deutschland GmbH (DE) 1999-04-14 EP disclosed