SCHEMBL324261

SCHEMBL324261

O=C(Oc1cccc(Cl)c1)N1C=Cc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.46
HSD17B3 P37058 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
TRPA1 O75762 2/20 0.41
FNTA P49354 2/20 0.37
FNTB P49356 2/20 0.37
FKBP1A P62942 1/20 0.35
HRH3 Q9Y5N1 3/20 0.35
OPRM1 P35372 1/20 0.35
NPC1 O15118 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
OGT O15294 1/20 0.34
KMT2A Q03164 1/20 0.34
EPHX1 P07099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL324821 0.85 SMN1; SMN2 (0.55) BCHEHSD17B3SMN1; SMN2NPC1RAB9A
SCHEMBL325206 0.80 HCAR2 (0.43) HSD17B3NPC1RAB9AKMT2A
SCHEMBL323656 0.78 BCHE (0.43) BCHEHSD17B3SMN1; SMN2NPC1CASP3
SCHEMBL324830 0.78 LIPE (0.44) BCHESMN1; SMN2NPC1CASP3RAB9A
SCHEMBL15055276 0.74 MGLL (0.46)
SCHEMBL324441 0.74 HSD17B3 (0.43) HSD17B3
SCHEMBL325232 0.74 HSD17B3 (0.46) HSD17B3
SCHEMBL323930 0.74 HSD17B3 (0.46) HSD17B3SMN1; SMN2KMT2A
SCHEMBL3628702 0.74 P2RX4 (0.46) BCHEHSD17B3SMN1; SMN2TRPA1KMT2A
SCHEMBL8573553 0.73 HSD17B3 (0.39) HSD17B3SMN1; SMN2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590944-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd. (CH) 2013-05-15 EP disclosed
US-20130109685-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD. (CH) 2013-05-02 US disclosed
WO-2012004722-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109685-A1 1-PHENYL-SUBSTITUTED HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS PTGER1, PTGDR, PTGDR2 BCHE 4335/4885HSD17B3 967/4885SMN1; SMN2 4056/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.