SCHEMBL3243076

SCHEMBL3243076

CC(O)c1ccc2c(c1)CCNC2

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 3/20 0.51
DRD2 P14416 1/20 0.49
DRD3 P35462 1/20 0.49
PNMT P11086 4/20 0.46
CD44 P16070 1/20 0.46
MAOB P27338 1/20 0.46
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
ADCY6 O43306 1/20 0.42
ADCY3 O60266 1/20 0.42
ADCY9 O60503 1/20 0.42
ADCY5 O95622 1/20 0.42
ADCY8 P40145 1/20 0.42
ADCY7 P51828 1/20 0.42
ADCY2 Q08462 1/20 0.42
ADCY1 Q08828 1/20 0.42
ADCY4 Q8NFM4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12608371 0.89 ADCY6 (0.50) DRD2DRD3ADCY6ADCY3ADCY9
SCHEMBL4565700 0.86 ASIC3 (0.55) ASIC3DRD2DRD3PNMTCD44
Hydrochloric Acid SCHEMBL1265678 0.84 ASIC3 (0.53) ASIC3DRD2DRD3PNMTCD44
Hydrochloric Acid SCHEMBL30297516 0.84 UGT2B7 (0.41)
SCHEMBL18717400 0.83 ASIC3 (0.51) ASIC3DRD2DRD3PNMTCD44
SCHEMBL3247113 0.83 ASIC3 (0.51) ASIC3DRD2DRD3PNMTCD44
SCHEMBL3055999 0.83 ASIC3 (0.51) ASIC3DRD2DRD3PNMTCD44
SCHEMBL17585071 0.82 ASIC3 (0.55) ASIC3DRD2DRD3PNMTCD44
SCHEMBL20510027 0.81 ASIC3 (0.46) ASIC3DRD2DRD3
SCHEMBL21118921 0.80 ASIC3 (0.49) ASIC3DRD2DRD3PNMTCD44

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021138498-A1 CD73 INHIBITOR AND A2A/A2B ADENOSINE RECEPTOR INHIBITOR COMBINATION THERAPY INCYTE CORPORATION (US) 2021-07-08 WO disclosed
WO-2010022055-A2 INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS AMGEN INC. (US) 2010-02-25 WO disclosed