SCHEMBL3243835

SCHEMBL3243835

Cc1c(-c2ccno2)sc(N2CCOCC2)c1C#Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
PIK3CA P42336 8/20 0.35
GRM5 P41594 5/20 0.35
AR P10275 1/20 0.35
MTOR P42345 3/20 0.35
PIK3R1 P27986 2/20 0.35
BRD4 O60885 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GRM4 Q14833 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119485 0.74 PIK3CA (0.48) PIK3CAGRM5PIK3R1BRD4PIK3CD
SCHEMBL3265059 0.73 PIK3CA (0.43) PIK3CAGRM5BRD4
SCHEMBL3121821 0.73 PIK3CA (0.44) PIK3CAGRM5NPC1RAB9A
SCHEMBL3130106 0.73 PIK3CA (0.48) PIK3CAGRM5PIK3R1BRD4PIK3CD
SCHEMBL16161774 0.70 GRM5 (0.46) PIK3CAGRM5PIK3R1BRD4PIK3CD
SCHEMBL3754871 0.70 PIK3CA (0.43) PIK3CAGRM5PIK3R1BRD4GRM4
SCHEMBL3120379 0.69 PIK3CA (0.41) PIK3CAGRM5NPC1
SCHEMBL3116360 0.69 GRM5 (0.50) PIK3CAGRM5MTORNPC1RAB9A
SCHEMBL3765027 0.68 BRD4 (0.36) PIK3CAGRM5PIK3R1BRD4GRM4
SCHEMBL16161712 0.67 HTT (0.47) PIK3CAGRM5PIK3R1BRD4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001126-A1 THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-01-07 WO disclosed