SCHEMBL3130106

SCHEMBL3130106

Cc1c(C(N)=O)sc(N2CCOCC2)c1C#Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.48
HSD17B10 Q99714 3/20 0.40
CHRNA7 P36544 2/20 0.40
BRD4 O60885 1/20 0.39
GRM5 P41594 5/20 0.39
CHRNA1 P02708 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR3A P46098 1/20 0.38
IKBKB O14920 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
PIK3CD O00329 2/20 0.37
PIK3CB P42338 2/20 0.37
PIK3CG P48736 1/20 0.37
ACACB O00763 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119485 0.91 PIK3CA (0.48) PIK3CAHSD17B10CHRNA7BRD4GRM5
SCHEMBL3265059 0.90 PIK3CA (0.43) PIK3CAHSD17B10CHRNA7BRD4GRM5
SCHEMBL3121821 0.89 PIK3CA (0.44) PIK3CAHSD17B10CHRNA7GRM5CHRNA1
SCHEMBL3120379 0.85 PIK3CA (0.41) PIK3CAHSD17B10CHRNA7GRM5CHRNA1
SCHEMBL3116360 0.84 GRM5 (0.50) PIK3CAHSD17B10GRM5KDM4EALDH1A1
SCHEMBL3425682 0.79 PIK3CA (0.61) PIK3CAIKBKBKDM4EALDH1A1GAA
SCHEMBL3268335 0.78 PIK3CA (0.42) PIK3CABRD4IKBKBKDM4EALDH1A1
SCHEMBL3247973 0.75 PIK3CA (0.47) PIK3CAHSD17B10IKBKBKDM4EALDH1A1
SCHEMBL3243835 0.73 PTGS2 (0.36) PIK3CABRD4GRM5PIK3CDPIK3CB
SCHEMBL3124602 0.71 HSD17B10 (0.51) PIK3CAHSD17B10CHRNA7BRD4GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001126-A1 THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-01-07 WO disclosed