SCHEMBL3265059

SCHEMBL3265059

CC(=O)c1sc(N2CCOCC2)c(C#Cc2ccccc2)c1C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.43
HSD17B10 Q99714 1/20 0.41
CHRNA7 P36544 2/20 0.41
GRM5 P41594 7/20 0.39
ACACB O00763 1/20 0.39
CHRNA1 P02708 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
HTR3A P46098 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
ALOX15 P16050 1/20 0.38
BRD4 O60885 1/20 0.38
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119485 0.92 PIK3CA (0.48) PIK3CAHSD17B10CHRNA7GRM5ACACB
SCHEMBL3130106 0.90 PIK3CA (0.48) PIK3CAHSD17B10CHRNA7GRM5ACACB
SCHEMBL3121821 0.90 PIK3CA (0.44) PIK3CAHSD17B10CHRNA7GRM5CHRNA1
SCHEMBL3120379 0.86 PIK3CA (0.41) PIK3CAHSD17B10CHRNA7GRM5CHRNA1
SCHEMBL3116360 0.85 GRM5 (0.50) PIK3CAHSD17B10GRM5ALDH1A1MAPT
SCHEMBL3124602 0.76 HSD17B10 (0.51) PIK3CAHSD17B10CHRNA7GRM5ACACB
SCHEMBL3264448 0.74 PIK3CA (0.48) PIK3CAHSD17B10CHRNA7ALDH1A1MAPT
SCHEMBL3243835 0.73 PTGS2 (0.36) PIK3CAGRM5BRD4
SCHEMBL3119056 0.72 PIK3CA (0.41) PIK3CAHSD17B10CHRNA7CHRNA1CHRNA3
SCHEMBL623321 0.71 PIK3CA (0.45) PIK3CAHSD17B10ACACBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001126-A1 THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-01-07 WO disclosed