SCHEMBL3244548

SCHEMBL3244548

COc1cc2c(c(OC)c1OC)C(CCCCC1c3c(cc(OC)c(OC)c3OC)CCN1C)N(C)CC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN2 Q9H2S1 4/20 0.60
KCNN3 Q9UGI6 4/20 0.60
KCNN1 Q92952 2/20 0.60
HTR2A P28223 6/20 0.51
HTR2C P28335 6/20 0.51
HTR7 P34969 6/20 0.51
HTR2B P41595 6/20 0.51
HTR1A P08908 5/20 0.51
DRD1 P21728 4/20 0.51
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
DRD2 P14416 3/20 0.51
TDP2 O95551 2/20 0.51
MAPT P10636 2/20 0.51
CASP3 P42574 2/20 0.51
RAD52 P43351 2/20 0.51
SENP8 Q96LD8 2/20 0.51
SENP7 Q9BQF6 2/20 0.51
SENP6 Q9GZR1 2/20 0.51
HSD17B10 Q99714 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3253192 0.99 KCNN2 (0.61) KCNN2KCNN3KCNN1HTR2AHTR2C
SCHEMBL3250383 0.97 KCNN2 (0.64) KCNN2KCNN3KCNN1HTR2AHTR2C
Hydrochloric Acid SCHEMBL3248244 0.96 KCNN2 (0.65) KCNN2KCNN3KCNN1HTR2AHTR2C
SCHEMBL4413729 0.84 LMNA (0.60) KCNN2KCNN3KCNN1DRD1KDM4E
SCHEMBL2112127 0.84 LMNA (0.60) KCNN2KCNN3KCNN1DRD1KDM4E
Hydrochloric Acid SCHEMBL10746848 0.83 LMNA (0.58) KCNN2KCNN3KCNN1DRD1KDM4E
Hydrochloric Acid SCHEMBL11099161 0.83 LMNA (0.58) KCNN2KCNN3KCNN1DRD1KDM4E
SCHEMBL6130855 0.79 HTR7 (0.52) HTR2AHTR2CHTR7HTR2BHTR1A
SCHEMBL6130831 0.79 HTR7 (0.52) HTR2AHTR2CHTR7HTR2BHTR1A
SCHEMBL3253219 0.78 KCNN2 (0.94) KCNN2KCNN3KCNN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1998775-B1 BIS1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USES AS PHARMACEUTICALS UNIV LIEGE (BE) 2010-05-19 EP claimed