SCHEMBL3244773

SCHEMBL3244773

CC(C)C(=O)Nc1cc(C2C[CH]C2)n[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA1 P30542 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 1/20 0.35
RECQL P46063 1/20 0.35
CDK2 P24941 4/20 0.34
CCNA2 P20248 3/20 0.34
CCNA1 P78396 3/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM5A P29375 1/20 0.34
PARP1 P09874 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK5 Q00535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1106976 0.88 CCNA2 (0.40) ALDH1A1LMNAHSD17B10ADORA1CDK2
SCHEMBL6388094 0.83 ALDH1A1 (0.34) ALDH1A1LMNAHSD17B10ADORA1SMN1; SMN2
SCHEMBL6388050 0.81 KDM5A (0.37) ALDH1A1LMNAHSD17B10ADORA1KDM4E
SCHEMBL6388056 0.81 KDM5A (0.37) ALDH1A1LMNAHSD17B10ADORA1KDM4E
SCHEMBL6388085 0.81 CDK2 (0.34) ALDH1A1LMNAHSD17B10ADORA1KDM4E
SCHEMBL6388090 0.81 CDK2 (0.34) ALDH1A1LMNAHSD17B10ADORA1KDM4E
SCHEMBL3260157 0.80 ADORA1 (0.39) ALDH1A1HSD17B10ADORA1SMN1; SMN2KDM4E
SCHEMBL6386568 0.78 ADORA1 (0.33) ALDH1A1LMNAHSD17B10ADORA1SMN1; SMN2
SCHEMBL6386570 0.78 ADORA1 (0.33) ALDH1A1LMNAHSD17B10ADORA1SMN1; SMN2
SCHEMBL3257731 0.78 L3MBTL1 (0.41) ALDH1A1LMNAHSD17B10ADORA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689721-B1 AMINOPYRAZOLE DERIVATIVES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2010-07-14 EP claimed