SCHEMBL3244881

SCHEMBL3244881

COc1ccc2c(c1)CN(C(=O)CN1C(=O)CCc3cc(Br)cnc31)C2

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
NAMPT P43490 5/20 0.38
TAAR1 Q96RJ0 1/20 0.36
ABHD6 Q9BV23 1/20 0.36
RYR2 Q92736 1/20 0.36
MGAT3 Q09327 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
TIPARP Q7Z3E1 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240895 0.94 TAAR1 (0.43) ESR1ESR2TAAR1ABHD6CYP2C19
SCHEMBL3119103 0.85 GAA (0.42) ROCK1ESR1ESR2NAMPTTIPARP
SCHEMBL3120168 0.83 TAAR1 (0.46) ESR1ESR2TAAR1CYP2C19
SCHEMBL3244879 0.83 LMNA (0.38)
SCHEMBL3247392 0.82 HSD17B3 (0.43) ROCK1ESR1ESR2NAMPT
SCHEMBL3128418 0.82 ROCK1 (0.37) ROCK1ESR1ESR2NAMPTTIPARP
SCHEMBL3239092 0.81 GRIN2B (0.43) ROCK1ESR1ESR2
SCHEMBL3131972 0.81 MAPT (0.42) ESR1ESR2TAAR1CYP2C19
SCHEMBL3126513 0.81 ESR2 (0.45) ESR1ESR2TAAR1ABHD6CYP2C19
SCHEMBL3122093 0.81 TAAR1 (0.46) ESR1ESR2TAAR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed