SCHEMBL3248554

SCHEMBL3248554

COc1ccc2c(c1)CN(C(=O)CN1C(=O)CCc3cc(-c4cncnc4)cnc31)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.41
ESR1 P03372 1/20 0.41
PORCN Q9H237 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
CYP11B2 P19099 5/20 0.40
CYP11B1 P15538 5/20 0.40
CHRM4 P08173 1/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
NR4A1 P22736 1/20 0.40
APEX1 P27695 1/20 0.40
RECQL P46063 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3246260 0.92 CYP11B1 (0.48) ESR2ESR1PORCNTAAR1CYP11B2
SCHEMBL3252487 0.91 CYP11B1 (0.51) ESR2ESR1PORCNTAAR1CYP11B2
SCHEMBL3119024 0.91 TAAR1 (0.46) ESR2ESR1PORCNTAAR1CYP11B1
SCHEMBL13521725 0.90 CYP11B1 (0.47) ESR2ESR1TAAR1CYP11B2CYP11B1
SCHEMBL3264528 0.89 MAPK1 (0.44) ESR2ESR1PORCNTAAR1CYP11B2
SCHEMBL3127545 0.89 MAPK1 (0.41) ESR2ESR1PORCNTAAR1CYP11B2
SCHEMBL3251460 0.88 CHRM4 (0.42) ESR2ESR1TAAR1CYP11B2CYP11B1
SCHEMBL3243098 0.88 GRIN2B (0.41) ESR2ESR1TAAR1CYP11B2CYP11B1
SCHEMBL13521598 0.87 HSD17B3 (0.43) ESR2ESR1TAAR1CYP11B2CYP11B1
SCHEMBL3120168 0.87 TAAR1 (0.46) ESR2ESR1TAAR1CHRM4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed