SCHEMBL3249334

SCHEMBL3249334

COc1ccc2c(c1)CN(C(=O)CN1CCOc3cc(Br)cnc31)CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
ESR2 Q92731 2/20 0.40
ESR1 P03372 1/20 0.40
MAPT P10636 6/20 0.40
TDP1 Q9NUW8 2/20 0.40
RIPK1 Q13546 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ABCB1 P08183 2/20 0.39
ABCC1 P33527 1/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
NR4A1 P22736 1/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
KMT2A Q03164 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249745 0.85 GAA (0.49) MAPK1TAAR1ESR2ESR1MAPT
SCHEMBL3240895 0.79 TAAR1 (0.43) MAPK1TAAR1ESR2ESR1MAPT
SCHEMBL3120660 0.78 GAA (0.49) MAPK1TAAR1MAPTTDP1GAA
SCHEMBL3119103 0.78 GAA (0.42) ESR2ESR1GAAALDH1A1SMN1; SMN2
SCHEMBL3237347 0.75 GAA (0.48) MAPK1MAPTTDP1GAAALDH1A1
SCHEMBL13521762 0.73 TAAR1 (0.41) TAAR1ESR2ESR1MAPTTDP1
SCHEMBL3241489 0.73 TSHR (0.46) MAPK1TAAR1ESR2ESR1MAPT
SCHEMBL3126815 0.73 GAA (0.51) MAPK1ESR2ESR1MAPTTDP1
SCHEMBL3252753 0.72 TSHR (0.44) MAPK1TAAR1ESR2ESR1MAPT
SCHEMBL13521636 0.72 TSHR (0.50) MAPK1TAAR1ESR2MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed