SCHEMBL3249728

SCHEMBL3249728

Cc1ccccc1-c1[c]c2ccccc2cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
CYP2A6 P11509 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
CYP1A2 P05177 4/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 2/20 0.33
DCUN1D1 Q96GG9 2/20 0.33
ACHE P22303 1/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
HPGD P15428 2/20 0.33
BRD4 O60885 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8178726 0.82 CYP2A6 (0.42) ALDH1A1CYP2A6NPC1RAB9ASMN1; SMN2
SCHEMBL8148539 0.82 CYP2A6 (0.42) ALDH1A1CYP2A6NPC1RAB9ASMN1; SMN2
SCHEMBL239122 0.79 CYP2A6 (0.37) ALDH1A1CYP2A6CYP1A2CYP3A4TSHR
SCHEMBL4609078 0.77 MAPK1 (0.39) ALDH1A1CYP2A6RAB9ASMN1; SMN2DCUN1D1
SCHEMBL3240933 0.77 CYP2A6 (0.39) ALDH1A1CYP2A6NPC1RAB9ASMN1; SMN2
SCHEMBL3246275 0.77 NPC1 (0.37) ALDH1A1NPC1RAB9ASMN1; SMN2CASP3
SCHEMBL668159 0.77 ALDH1A1 (0.41) ALDH1A1CYP2A6SMN1; SMN2CYP1A2CYP3A4
SCHEMBL10501303 0.77 ALDH1A1 (0.39) ALDH1A1NPC1RAB9ASMN1; SMN2CASP3
SCHEMBL667984 0.77 ALDH1A1 (0.34) ALDH1A1CYP2A6RAB9ASMN1; SMN2TSHR
SCHEMBL3241635 0.77 ALDH1A1 (0.44) ALDH1A1NPC1RAB9ASMN1; SMN2DCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1167366-B1 AMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2010-05-05 EP disclosed
EP-1473297-B1 PROCESS FOR PRODUCING TERTIARY PHOSPHINE HAVING BULKY HYDROCARBON GROUP BONDED HOKKO CHEM IND CO (JP) 2009-10-14 EP disclosed
WO-2008091594-A2 FUNGICIDAL MIXTURES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-31 WO disclosed
EP-1948649-A2 FUNGICIDAL CARBOXAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-30 EP disclosed
US-7250535-B2 Process for producing tertiary phosphine HOKKO CHEMICAL INDUSTRY CO., LTD. (JP) 2007-07-31 US disclosed
WO-2007014290-A2 FUNGICIDAL CARBOXAMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2007-02-01 WO disclosed
US-20060020148-A1 Process for producing tertiary phosphine having bulky hydrocarbon group bonded HOLLO CHEMICAL INDUSTRY CO., LTD (JP) 2006-01-26 US disclosed
EP-1473297-A1 PROCESS FOR PRODUCING TERTIARY PHOSPHINE HAVING BULKY HYDROCARBON GROUP BONDED HOKKO CHEMICAL INDUSTRY CO. LTD. (JP) 2004-11-03 EP disclosed
US-6562849-B1 Amine compound or pharmacologically acceptable salt thereof. These compounds are useful in the treatment and/or prophylaxis of diseases such as diabetes, hyperlipemia, arteriosclerosis, cancer, etc. SANKYO COMPANY, LIMITED (JP) 2003-05-13 US disclosed
US-20030078426-A1 Amine derivative compounds SANKYO COMPANY, LIMITED (JP) 2003-04-24 US disclosed
EP-1167366-A1 AMINE DERIVATIVES Sankyo Company, Limited (JP) 2002-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060020148-A1 Process for producing tertiary phosphine having bulky hydrocarbon group bonded HRH3, HRH4, HRH1 ALDH1A1 1764/4885CYP2A6 2988/4885NPC1 4180/4885
US-20030078426-A1 Amine derivative compounds H1-10, APOB, PRMT1 ALDH1A1 874/4885CYP2A6 2385/4885NPC1 359/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.