SCHEMBL3250445

SCHEMBL3250445

CN(C)C(=O)c1cc(-c2cn[nH]c2)ccc1NC(=O)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.63
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ROCK1 Q13464 7/20 0.44
MYLK4 Q86YV6 2/20 0.44
MGLL Q99685 1/20 0.44
TACR3 P29371 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249281 0.89 ROCK2 (0.55) ROCK2NPC1RAB9AROCK1
SCHEMBL3241665 0.85 ROCK2 (0.69) ROCK2ROCK1
SCHEMBL3239730 0.82 ROCK2 (0.59) ROCK2NPC1RAB9AROCK1
SCHEMBL3250291 0.82 ROCK2 (0.74) ROCK2NPC1RAB9AROCK1
SCHEMBL3255236 0.82 NPC1 (0.46) ROCK2NPC1RAB9AMGLLTACR3
SCHEMBL13391233 0.82 ROCK2 (0.72) ROCK2ROCK1
SCHEMBL3241298 0.81 ROCK2 (0.55) ROCK2NPC1RAB9AROCK1MYLK4
SCHEMBL3244746 0.81 ROCK2 (0.57) ROCK2ROCK1
SCHEMBL3241905 0.80 ROCK2 (0.60) ROCK2ROCK1
SCHEMBL3248274 0.78 ROCK2 (1.00) ROCK2ROCK1MYLK4MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed