SCHEMBL3255236

SCHEMBL3255236

Cc1n[nH]cc1-c1ccc(NC(=O)OCc2ccccc2)c(C(=O)N(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ROCK2 O75116 1/20 0.43
PARP1 P09874 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAF1 P04049 1/20 0.41
BRAF P15056 1/20 0.41
CASP3 P42574 2/20 0.40
MGLL Q99685 3/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
TACR3 P29371 1/20 0.39
BRD4 O60885 1/20 0.39
FAAH O00519 1/20 0.39
BTK Q06187 2/20 0.39
POLB P06746 1/20 0.39
ENPP2 Q13822 1/20 0.39
MAOB P27338 1/20 0.39
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13390958 0.82 ROCK2 (0.51) NPC1RAB9AROCK2BTK
SCHEMBL3250445 0.82 ROCK2 (0.63) NPC1RAB9AROCK2MGLLTACR3
SCHEMBL3242948 0.80 ROCK2 (0.62) NPC1RAB9AROCK2SMN1; SMN2MGLL
SCHEMBL3249281 0.72 ROCK2 (0.55) NPC1RAB9AROCK2
SCHEMBL3238410 0.70 ROCK2 (0.64) NPC1RAB9AROCK2SMN1; SMN2MGLL
SCHEMBL6187342 0.69 NPC1 (0.52) NPC1RAB9ASMN1; SMN2RAF1BRAF
SCHEMBL6166293 0.68 PTPN1 (0.61) NPC1RAB9AROCK2MGLLHDAC3
SCHEMBL6189531 0.68 TACR3 (0.53) NPC1RAB9ACASP3MGLLTACR3
SCHEMBL3241665 0.67 ROCK2 (0.69) ROCK2
SCHEMBL6161722 0.67 MGLL (0.56) NPC1RAB9ASMN1; SMN2CASP3MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed