SCHEMBL3255804

SCHEMBL3255804

CC(C)(C)OC(=O)NCCNCc1nc2ccccc2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.50
HPGD P15428 3/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 2/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
BRD4 O60885 1/20 0.44
MAPT P10636 3/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4159541 0.89 HPGD (0.55) BCHEHPGDCYP1A2CYP2C19HTT
SCHEMBL1981436 0.81 BCHE (0.58) BCHECYP1A2CYP2C19HTTHDAC3
SCHEMBL3250296 0.77 MAPT (0.53) HPGDCYP1A2CYP2C19HTTMAPT
SCHEMBL25955151 0.75 HDAC3 (0.49) HPGDCYP1A2CYP2C19HTTHDAC3
SCHEMBL28366491 0.75 DYRK1A (0.48) HPGDRAB9AL3MBTL1SMN1; SMN2NPC1
SCHEMBL30493007 0.75 DYRK1A (0.48) HPGDRAB9AL3MBTL1SMN1; SMN2NPC1
SCHEMBL15195148 0.75 HPGD (0.58) HPGDCYP1A2CYP2C19HTTMAPT
SCHEMBL13539033 0.75 SMN1; SMN2 (0.63) HPGDCYP1A2CYP2C19HTTMAPT
SCHEMBL5068294 0.75 ALDH1A1 (0.53) BCHEHPGDHDAC3HDAC4HDAC1
SCHEMBL22605044 0.74 ATM (0.58) BCHEKMT2AKDM4EMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed