SCHEMBL3257705

SCHEMBL3257705

Cc1cc(CCC(=O)N2CCN(c3nccs3)CC2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.43
ME2 P23368 3/20 0.43
ME1 P48163 3/20 0.43
ME3 Q16798 3/20 0.43
SLC6A7 Q99884 1/20 0.43
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PARP1 P09874 1/20 0.42
GRM5 P41594 2/20 0.41
GRM1 Q13255 1/20 0.41
GFER P55789 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
AOC3 Q16853 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5179616 0.90 SLC6A7 (0.45) SCDME2ME1ME3SLC6A7
SCHEMBL3259324 0.83 ALDH1A1 (0.48) SCDME2ME1ME3SLC6A7
SCHEMBL5178153 0.80 ME2 (0.61) ME2ME1ME3KMT2AALDH1A1
SCHEMBL3257527 0.76 ALDH1A1 (0.46) SCDME2ME1ME3SLC6A7
SCHEMBL3151726 0.75 SCD (0.43) SCDSLC6A7PARP1GRM5GRM1
SCHEMBL15002301 0.74 GRM5 (0.53) SCDSLC6A7GRM5KDM4ETP53
SCHEMBL15002298 0.74 GRM5 (0.47) SLC6A7KMT2AALDH1A1GRM5KDM4E
SCHEMBL5178383 0.73 GRM5 (0.54) SCDSLC6A7KMT2AALDH1A1GRM5
SCHEMBL14340911 0.73 SCD (0.49) SCDSLC6A7ALDH1A1GRM5GRM1
SCHEMBL11080726 0.71 SLC6A7 (0.53) SCDSLC6A7KMT2AALDH1A1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765816-B1 SUBSTITUTED 1-PROPIOLYLPIPERAZINES HAVING AN AFFINITY FOR THE MGLUR5 RECEPTOR IN ORDER TO TREAT PAINFUL CONDITIONS GRUENENTHAL GMBH (DE) 2010-03-10 EP disclosed