SCHEMBL3258564

SCHEMBL3258564

OCC1Cc2cc(Cl)ccc2N1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 15/20 0.51
TRPM4 Q8TD43 8/20 0.51
CREBBP Q92793 1/20 0.41
PNMT P11086 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6194447 0.83 TRPM5 (0.43) TRPM5TRPM4
SCHEMBL19098966 0.81 PNMT (0.61) CREBBPPNMT
SCHEMBL471068 0.79 TRPM5 (0.51) TRPM5TRPM4
SCHEMBL7297572 0.76 PDE3B (0.41) CREBBPPNMT
SCHEMBL7297564 0.76 PDE3B (0.41) CREBBPPNMT
SCHEMBL2450511 0.74 CREBBP (0.59) TRPM5CREBBPPNMT
SCHEMBL1193549 0.74 CREBBP (0.59) TRPM5CREBBPPNMT
SCHEMBL30681442 0.74 CREBBP (0.59) TRPM5CREBBPPNMT
SCHEMBL550431 0.74 CREBBP (0.59) TRPM5CREBBPPNMT
SCHEMBL30288510 0.74 CREBBP (0.59) TRPM5CREBBPPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1330454-B1 BENZOPYRANYL HETEROCYCLE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DONGBU HITEK CO LTD (KR) 2010-05-19 EP disclosed
EP-1330454-A4 BENZOPYRANYL HETEROCYCLE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DONGBU HANNONG CHEMICAL CO LTD (KR) 2008-03-19 EP disclosed
EP-1330454-A1 BENZOPYRANYL HETEROCYCLE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dongbu Hannong Chemical Co., Ltd. (KR) 2003-07-30 EP disclosed
US-6413983-B1 COUPLING EPOXIDE WITH INDOLE OR QUINOLINE COMPOUND; PROTECT-ING HEART, BRAIN, RETINA AND NEURONAL CELL FROM ?ISCHEMIA-REPERFUSION? INJURY; SUPPRESSING LIPID PEROXIDATION DONGBU HANNONG CHEMICAL CO. LTD. (KR) 2002-07-02 US disclosed
WO-2002030925-A1 BENZOPYRANYL HETEROCYCLE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DONGBU HANNONG CHEMICAL CO., LTD (KR) 2002-04-18 WO disclosed