SCHEMBL550431

SCHEMBL550431

OCC1Cc2ccccc2N1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 1/20 0.59
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
PRKCD Q05655 6/20 0.44
PRKCG P05129 1/20 0.44
PRKCA P17252 1/20 0.44
PNMT P11086 4/20 0.41
MTNR1A P48039 3/20 0.41
TRPM5 Q9NZQ8 1/20 0.40
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2450511 1.00 CREBBP (0.59) CREBBPGAAMAPTPRKCDPRKCG
SCHEMBL29427458 1.00 CREBBP (0.59) CREBBPGAAMAPTPRKCDPRKCG
SCHEMBL30681442 1.00 CREBBP (0.59) CREBBPGAAMAPTPRKCDPRKCG
SCHEMBL30288510 1.00 CREBBP (0.59) CREBBPGAAMAPTPRKCDPRKCG
SCHEMBL1193549 1.00 CREBBP (0.59) CREBBPGAAMAPTPRKCDPRKCG
SCHEMBL16671960 0.85 GAA (0.47) CREBBPGAAMAPTPNMTMTNR1A
SCHEMBL11319601 0.85 GAA (0.47) CREBBPGAAMAPTPNMTMTNR1A
SCHEMBL14881136 0.82 PNMT (0.47) CREBBPGAAMAPTPNMTMTNR1A
SCHEMBL11426860 0.82 GAA (0.47) CREBBPGAAMAPTPNMTMTNR1A
SCHEMBL3441906 0.81 MTNR1A (0.56) CREBBPGAAMAPTPRKCDPRKCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 203 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586170-B Indolinyl acyl derivative and synthetic method of isoquinoline formyl derivative 江苏集萃分子工程研究院有限公司 2024-04-09 CN claimed
CN-117586170-A Indolinyl acyl derivative and synthetic method of isoquinoline formyl derivative 江苏集萃分子工程研究院有限公司 2024-02-23 CN claimed
CN-110279121-A A kind of Oligopeptide Compositions and preparation method thereof 海盐县凌特生物科技有限公司 2019-09-27 CN claimed
EP-2470508-A1 CANNABINOID RECEPTOR MODULATORS Arena Pharmaceuticals, Inc. (US) 2012-07-04 EP claimed
WO-2011025541-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. (US) 2011-03-03 WO claimed
CN-101657457-A Be used to prepare 1,3, the method for 2-oxa-boron acridine compound ZACH SYSTEM FR 2010-02-24 CN claimed
US-7586015-B2 Process for the preparation of 1,3,2-oxazaborolidine compounds ZACH SYSTEM (FR) 2009-09-08 US claimed
US-20080139851-A1 R2, R3, R4 and R5 are especially a hydrogen atom or an alkyl,wherein the following are reacted in two steps:a) a boric precursor compound with an acetal compound to give a boronate compound; and) the boronate compound with an amino alcohol compound PPG-SIPSY (FR) 2008-06-12 US claimed
US-12516053-B2 Bcl-2 inhibitors BEONE MEDICINES I GMBH (CH) 2026-01-06 US disclosed
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS AG (CH) 2025-05-29 US disclosed
US-12312349-B2 Apoptosis-inducing agents FOCHON PHARMACEUTICALS, LTD. (CN) 2025-05-27 US disclosed
EP-4540240-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME Monte Rosa Therapeutics AG (CH) 2025-04-23 EP disclosed
WO-2024201248-A1 COMPOUNDS AND METHODS FOR DEGRADING GSPT1 PIN THERAPEUTICS, INC. (KR) 2024-10-03 WO disclosed
WO-2024120471-A1 COMPOUNDS TARGETING MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-06-13 WO disclosed
EP-0642508-A1 TRICYCLIC QUINOXALINEDIONES AS GLUTAMATE RECEPTOR ANTAGONISTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1995-03-15 EP disclosed
CN-1094038-A The amino pyrazoles that replaces PFIZER (US) 1994-10-26 CN disclosed
WO-1994013644-A1 AMINO-SUBSTITUTED PYRAZOLES HAVING CRF ANTAGONISTIC ACTIVITY PFIZER INC. (US) 1994-06-23 WO disclosed
WO-1993008188-A1 TRICYCLIC QUINOXALINEDIONES AS GLUTAMATE RECEPTOR ANTAGONISTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1993-04-29 WO disclosed
US-4260628-A 2-Guanidinomethyl-indolines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-04-07 US disclosed
US-4153699-A ANALGESIC, ANTIPYRETIC, ANTIINFLAMMATORY RHONE-POULENC INDUSTRIES (FR) 1979-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080139851-A1 R2, R3, R4 and R5 are especially a hydrogen atom or an alkyl,wherein the following are reacted in two steps:a) a boric precursor compound with an acetal compound to give a boronate compound; and) the boronate compound with an amino alcohol compound ADH1A, ADH1C, ADH5 CREBBP 1036/4885GAA 4784/4885MAPT 3759/4885
US-12312349-B2 Apoptosis-inducing agents BCL2, BAX, BAD CREBBP 116/4885GAA 2247/4885MAPT 3573/4885
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME PSMA1, CSNK1G1, CSNK1A1 CREBBP 2136/4885GAA 234/4885MAPT 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.