SCHEMBL3261501

SCHEMBL3261501

CC1(C)OB(c2ccc3ncc(=O)[nH]c3c2)OC1(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
MAPKAPK2 P49137 1/20 0.40
RPS6KA3 P51812 1/20 0.40
CSNK2A1 P68400 1/20 0.40
PLK3 Q9H4B4 1/20 0.40
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
EGFR P00533 2/20 0.37
LPL P06858 5/20 0.36
LIPG Q9Y5X9 5/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3260516 0.89 MAPKAPK2 (0.50) ALDH1A1MAPKAPK2RPS6KA3CSNK2A1PLK3
SCHEMBL29490757 0.77 LPL (0.44) LPLLIPGPRMT5WDR77CA1
SCHEMBL874992 0.77 MMP12 (0.45) EGFRLPLLIPGSNCA
SCHEMBL2172654 0.77 LPL (0.44) LPLLIPGPRMT5WDR77CA1
SCHEMBL29525463 0.77 MMP12 (0.45) EGFRLPLLIPGSNCA
SCHEMBL15574354 0.75 ALDH1A1 (0.49) ALDH1A1IDO1TDO2LPLLIPG
SCHEMBL15296449 0.74 EGFR (0.40) ALDH1A1IDO1TDO2EGFRLPL
SCHEMBL3831957 0.74 PLAU (0.47) ALDH1A1IDO1TDO2EGFRLPL
SCHEMBL1226551 0.73 LPL (0.42) LPLLIPGPRMT5WDR77CA1
SCHEMBL2098959 0.72 CA9 (0.50) LPLLIPGCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020366-A1 AZABICYCLIC SUBSTITUTED 5-AMINOPYRAZOLES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed