SCHEMBL3263775

SCHEMBL3263775

COC(=O)c1cccnc1-c1c(C)c2ccccc2n1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAP2K1 Q02750 1/20 0.43
NR4A2 P43354 3/20 0.42
TSHR P16473 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 3/20 0.41
THRB P10828 1/20 0.41
MEN1 O00255 2/20 0.40
POLB P06746 1/20 0.40
IDO1 P14902 2/20 0.40
ALOX5AP P20292 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3857449 0.76 TDP1 (0.45) KDM4ETDP1NR4A2L3MBTL1PKM
SCHEMBL812065 0.74 KDM4E (0.59) KDM4ETDP1MAP2K1TSHRL3MBTL1
Tert-Butyl Formate SCHEMBL28781508 0.73 MAP2K1 (0.41) KDM4ETDP1MAP2K1NR4A2TSHR
SCHEMBL7649536 0.73 TDP1 (0.59) KDM4ETDP1MAP2K1TSHRL3MBTL1
SCHEMBL12166081 0.73 KDM4E (0.52) KDM4ETDP1MAP2K1NR4A2L3MBTL1
SCHEMBL31668450 0.70 ALDH1A1 (0.54) KDM4ETDP1TSHRL3MBTL1ALDH1A1
SCHEMBL27504693 0.70 ALDH1A1 (0.54) KDM4ETDP1TSHRL3MBTL1ALDH1A1
SCHEMBL28120694 0.69 TDP1 (0.50) KDM4ETDP1MAP2K1TSHRL3MBTL1
SCHEMBL29664560 0.69 TDP1 (0.54) KDM4ETDP1MAP2K1TSHRL3MBTL1
SCHEMBL645854 0.69 TDP1 (0.54) KDM4ETDP1MAP2K1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102204-B1 NEW AMINOPYRROLO[1,2- A]INDOLE ET AMINOPYRIDAZINO[1,6-A]INDOLE DERIVATIVES, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SERVIER LAB (FR) 2010-05-05 EP disclosed