SCHEMBL3264448

SCHEMBL3264448

CC(=O)c1sc(N2CCOCC2)c(C(=O)O)c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.48
PIK3CD O00329 1/20 0.48
PIK3CB P42338 1/20 0.48
ABCC1 P33527 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 2/20 0.41
POLB P06746 4/20 0.40
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GAA P10253 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3247973 0.87 PIK3CA (0.47) PIK3CAPIK3CDPIK3CBABCC1HTT
SCHEMBL3119056 0.82 PIK3CA (0.41) PIK3CAPIK3CDPIK3CBHSD17B10POLB
SCHEMBL3265059 0.74 PIK3CA (0.43) PIK3CAHTTHSD17B10ALDH1A1GAA
SCHEMBL18802958 0.71 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBHSD17B10ALDH1A1
SCHEMBL18412843 0.68 ALDH1A1 (0.51) PIK3CAPIK3CDPIK3CBHTTHSD17B10
SCHEMBL3121805 0.68 PRKDC (0.48) PIK3CAPIK3CDPIK3CBALDH1A1KDM4E
SCHEMBL18412822 0.68 PIK3CA (0.46) PIK3CAPIK3CDPIK3CBHTTHSD17B10
SCHEMBL1574758 0.68 PIK3CD (0.78) PIK3CAPIK3CDPIK3CBHTTALDH1A1
SCHEMBL21755209 0.68 PIK3CA (0.52) PIK3CAPIK3CDPIK3CBHTTHSD17B10
SCHEMBL3119485 0.67 PIK3CA (0.48) PIK3CAPIK3CDPIK3CBHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001126-A1 THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-01-07 WO disclosed