SCHEMBL3264462

SCHEMBL3264462

CN1C[C@H](O)C[C@H]1C(=O)N1CCN(Cc2cccc3cc(C(=O)O)n(C)c23)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FAAH O00519 5/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MCL1 Q07820 2/20 0.34
DHODH Q02127 2/20 0.34
RORC P51449 2/20 0.34
HRH3 Q9Y5N1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3264483 1.00 FAAH (0.35) FAAHMEN1KMT2AMCL1DHODH
SCHEMBL3266877 1.00 FAAH (0.35) FAAHMEN1KMT2AMCL1DHODH
SCHEMBL3232196 1.00 FAAH (0.35) FAAHMEN1KMT2AMCL1DHODH
SCHEMBL3267299 0.88 HRH3 (0.37) FAAHMEN1KMT2AHRH3KDM4E
SCHEMBL3232200 0.87 FAAH (0.34) FAAHMEN1KMT2ADHODHRORC
SCHEMBL3264487 0.87 FAAH (0.34) FAAHMEN1KMT2ADHODHRORC
SCHEMBL3266879 0.87 FAAH (0.34) FAAHMEN1KMT2ADHODHRORC
SCHEMBL3264465 0.87 FAAH (0.34) FAAHMEN1KMT2ADHODHRORC
SCHEMBL3267160 0.86 FAAH (0.38) FAAHMEN1KMT2AMCL1DHODH
SCHEMBL690572 0.85 RORC (0.40) FAAHMEN1KMT2AMCL1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010026096-A1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO claimed
WO-2010026096-A1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO disclosed